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March 5, 2015

Bronchial asthma drugs classification

Classification of Bronchial Asthma Drugs.

1)Bronchodilators : Relive Bronchospasm
2) Anti-inflammatory drugs : Prevent Bronchospasm

1)Bronchodilators : Relive Bronchospasm.

A. Adrenergic Drugs.
B. Antichoilnergic Drugs.
C. Methyl – xanthenes.

A. Adrenergic Drugs.

i. Non – selective.
ii. Selective β2 – agonists.

i. Non – selective.
  • Adrenaline
  • Isoprenaline
  • Ephedrine

ii. Selective β2 – agonists.
  • Salbutamol
  • Terbutaline
  • Bambuterol
  •  Fenoterol 
  •  Salmeterol
  •  Formeterol

B. Antichoilnergic Drugs :

  • Ipratropium
  • Tiotropium

C. Methyl – xanthenes.

  • Theophylline (anhydrous )
  • Aminophylline
  • Hydroxyethyl theophyline
  • Choline theophyllinate
  • Theophylline ethanolate or Piperazine
  • Doxophylline
  • Diprophylline

2. Anti – inflammatory drugs : Prevent Bronchospasm

A.Corticosteroids
B. Mast Cell Stabilizers
C. Anti-leukotriene Drugs
D. Anti – IgE antibodies

A. Corticosteroids :-

i. Inhalational :
  •  Bechomethasone
  • Triamcinolone
  • Budesonide
  •  Fluticasone
  •  Flunisolide
  • Ciclesonide
ii. Systemic :
  • Prednisolone
  • Hydrocortisone

B. Mast cell Stabilizers :

  • Sod. Cromoglycate
  • Nedocromyl
  • Ketotifen

C. Anti-leukotriens Drugs :-

i. Leukotriene synthesis inhibitor :
  •  Zileuton
ii. Leukotriene receptor antagonists :
  • Montelukast
  • Zafirlukast
  • Pranlukast
  • Iralukast
iii. Anti-IgE antibodies :
  • Omalizumab













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